AI drug discoveryConcept
PHGDH inhibitor series — seeking in vivo validation partner
[Demo post] We have a validated series of small-molecule PHGDH inhibitors with sub-micromolar potency in serine-dependent breast cancer lines, plus full SAR and selectivity data. We are looking for a group with orthotopic xenograft capability to take the lead compounds into an in vivo efficacy study.
Offering
Validated inhibitor seriesSAR dataset
Seeking
Co-investigator for R01
Karthikeya Thimirishetty · University of Alabama Birmingham